Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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1,666
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1,666
Tocris Bioscience™ NRX 252114
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Molecular glue Degrader of mutant β-catenin
| Target | Molecular Glues |
|---|---|
| CAS | 2763260-39-3 |
| Purity | 0.98 |
| Chemical Name or Material | 2-[[4-[(2,6-Dichlorophenyl)thio]-1,2-dihydro-2-oxo-6-(trifluoromethyl)-3-pyridinyl]carbonyl]-2,3-dihydro-1H-isoindole-4-carbonitrile |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C22H12Cl2F3N3O2S |
1,668
Tocris Bioscience™ DIM-C-pPhOH
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Nur77 antagonist
| CAS | 151358-47-3 |
|---|---|
| Chemical Name or Material | 1,1-Bis(3'-indolyl)-1-(p-hydroxyphenyl)methane |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C23H18N2O |
| Formula Weight | Observed MW: 338.408 |
| Assay Percent Range | >98% |
1,669
Tocris Bioscience™ BI 78D3
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CAS: 883065-90-5 Molecular Formula: C13H9N5O5S2
| CAS | 883065-90-5 |
|---|---|
| Molecular Formula | C13H9N5O5S2 |
1,670
Tocris Bioscience™ Cinacalcet hydrochloride
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Low molecular weight, organic compound that may help regulate biological process.
| Target | Calcium-Sensing Receptor |
|---|---|
| CAS | 364782-34-3 |
| Product Type | Inhibitor |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C22H22F3N.HCl |
| Formula Weight | 393.87g/mol |
1,671
Tocris Bioscience™ Trametinib
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Potent and selective MEK inhibitor; orally bioavailable
| Target | MEK Inhibitors |
|---|---|
| CAS | 871700-17-3 |
| Purity | 0.98 |
| Chemical Name or Material | N-[3-[3-Cyclopropyl-5-[(2-fluoro-4-iodophenyl)amino]-3,4,6,7-tetrahydro-6,8-dimethyl-2,4,7-trioxopyrido[4,3-d]pyrimidin-1(2 H)-yl]phenyl]acetamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C26H23FIN5O4 |
1,672
Tocris Bioscience™ Fludarabine
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CAS: 21679-14-1 Molecular Formula: C10H12FN5O4
| CAS | 21679-14-1 |
|---|---|
| Molecular Formula | C10H12FN5O4 |
1,673
Tocris Bioscience™ SK 216
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Plasminogen activator inhibitor-1 (PAI-1) inhibitor
| CAS | 654080-03-2 |
|---|---|
| Chemical Name or Material | 2-[5-[[6-[5-(1,1-Dimethylethyl)-2-benzoxazolyl]-2-naphthalenyl]oxy]pentyl]propanedioic acid disodium salt |
| Recommended Storage | Desiccate at Room Temperature |
| Molecular Formula | C29H29NO6Na2 |
| Formula Weight | Observed MW: 533.52 |
| Assay Percent Range | >98% |
1,674
Tocris Bioscience™ Ivosidenib
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Potent inhibitor of mutant isocitrate dehydrogenase (mIDH1)
| Target | Isocitrate Dehydrogenase 1/IDH1 |
|---|---|
| CAS | 1448347-49-6 |
| Chemical Name or Material | (2S)-N-{(1S)-1-(2-Chlorophenyl)-2-[(3,3-difluorocyclobutyl)amino]-2-oxoethyl}-1(4-cyanopyridin-2-yl)-N-(5-fluoropyridin-3-yl)-5-oxopyrrolidine-2-carboxamide |
| Recommended Storage | Store the unopened product at -20 to -70 °C. Use a manual defrost freezer and avoid repeated freeze-thaw cycles. Do not use past expiration date. |
| Molecular Formula | C28H22ClF3N6O3 |
1,675
Tocris Bioscience™ A 939572
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Potent SCD-1 inhibitor
| Target | Compounds for Stem Cell Differentiation |
|---|---|
| CAS | 1032229-3-6 |
| Purity | >99% |
| Chemical Name or Material | 4-(2-Chlorophenoxy)-N-[3-[(methylamino)carbonyl]phenyl]-1-piperidinecarboxamide |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C20H22ClN3O3 |
| Formula Weight | 387.86 |
1,676
Tocris Bioscience™ BIX 01294
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CAS: 1392399-03-9 Molecular Formula: C28H41Cl3N6O2
| CAS | 1392399-03-9 |
|---|---|
| Molecular Formula | C28H41Cl3N6O2 |
1,677
Tocris Bioscience™ FPS ZM1
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High affinity antagonist of RAGE
| CAS | 945714-67-0 |
|---|---|
| Chemical Name or Material | 4-Chloro-N-cyclohexyl-N-(phenylmethyl)benzamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C20H22ClNO |
| Formula Weight | Observed MW: 327.85 |
| Assay Percent Range | >99% |
1,678
Tocris Bioscience™ FAK Inhibitor 14
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CAS: 4506-66-5 Molecular Formula: C6H14Cl4N4
| CAS | 4506-66-5 |
|---|---|
| Molecular Formula | C6H14Cl4N4 |
1,680
Tocris Bioscience™ PluriSln 1
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CAS: 91396-88-2 Molecular Formula: C12H11N3O
| CAS | 91396-88-2 |
|---|---|
| Molecular Formula | C12H11N3O |